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“Systemic” therapies by biologic domain in advanced Prostate Cancer




                                   ‘Enhanced’                                                                                                      Targeted Agents
                              Androgen signaling   Chemotherapy                               Immunotherapy                Radioligand                 Precision
                                                                                                                              Agents
                                    inhibition                                                                                                          Therapy



                             Abiraterone Acetate                                              Sipuleucel T
                                Enzalutamide                    Docetaxel                      Pembrolizumab           Radium-223                     Olaparib
                                 Apalutamide                  Cabazitaxel                                                 Lu-PSMA                   Rucaparib
                                Darolutamide
                                   Abi + Apa                                                                                                       Ipatasertib












                                                                       Treatment of Primary


                                                           A systemic (equivalent) therapy ?


                            Source: Personal File




                                                                                                  Grey Listings: phase III data but no indication (yet)
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